Methenolone is a synthetic androgen and anabolic steroid. It is an agonist of the androgen receptor (AR), the biological target of androgens like testosterone and dihydrotestosterone (DHT). It exhibits moderate anabolic effects and weak androgenic effects, making it suitable for specific therapeutic applications.

Indications

• Strength Increase: Methenolone has the ability to enhance strength without significantly increasing muscular bulk, which is beneficial for athletes who are not bodybuilders.
• Muscular Endurance: Promotes increased muscular endurance and faster recovery.
• Fat Burning: Assists in increasing metabolic rate, making it an effective fat burner.

Contraindications

• Not intended for use in children.
• Known or suspected prostatic carcinoma and mammary carcinoma in males.
• Not intended for use in female patients other than those with disseminated breast cancer.
• Contraindicated in cases of nephrosis or the nephrotic phase of nephritis, cardiac and renal failure, hypercalcaemia, oedema, jaundice, liver disease with impaired bilirubin excretion, and testicular and hepatic carcinoma.

Dosage and Directions for Use

• Administration: Primobolic should be administered by deep intramuscular injection.
• Adult Dose: 50-100 mg every 3 weeks.

Side Effects and Special Precautions

• Virilization: This can appear in sensitive women as hoarseness, acne, hirsutism, and increased libido; in prepubertal boys as an increased frequency of erections and phallic enlargement, and in girls as an increase of pubic hair and clitoral hypertrophy. Hoarseness may be the first symptom of vocal change, which may end in a long-lasting, sometimes irreversible deepening of the voice.
• Other Adverse Reactions:
  • Oligospermia and decreased ejaculatory volume.
  • Suppression of ovarian activity, atrophy of the breasts and endometrial tissue.
  • Amenorrhoea and inhibition of spermatogenesis.
  • Water and salt retention.
  • Premature epiphyseal closure.
  • Increased nitrogen retention and skeletal weight.
  • Oedema.
  • Increased vascularity of the skin.
  • Increased growth of the bone.
  • Elderly males may become over-stimulated.

Monitoring

Patients with the following conditions should be monitored:

• Latent or overt cardiac failure, renal dysfunction, hypertension, epilepsy or migraine (or a history of these conditions), as anabolic steroids may induce salt and fluid retention.
• Diabetes, since anabolic steroids may improve glucose tolerance and decrease the need for insulin or other antidiabetic drugs.
• Incomplete statural growth, as anabolic steroids in high dosages may accelerate epiphyseal closure.
• Skeletal metastases, as anabolic steroids may induce hypercalcaemia and hypercalciuria in these patients.
• Liver dysfunction.

Interactions

Liver-enzyme-inducing agents may reduce the effects of Methenolone by enhancing its metabolism in the liver.

Storage

• Store at controlled room temperatures below 30°C and protect from light.
• If expired or damaged, return to your pharmacist for disposal.

Caution

Abuse of this product in sports is highly discouraged. Cooper Pharma does not take any responsibility for the use of this product for any other purpose. This product should be used under proper medical supervision.

Safety Information

• Keep out of the reach and sight of children.